Structure-activity relationship for the first-in-class clinical steroid sulfatase inhibitor Irosustat (STX64, BN83495).

Authors:
Woo LW; Ganeshapillai D; Thomas MP; Sutcliffe OB; Malini B and 3 more

Journal:
ChemMedChem

Publication Year: 2011

DOI:
10.1002/cmdc.201100288

PMCID:
PMC3262147

PMID:
21990014

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Journal Information

Full Title: ChemMedChem

Abbreviation: ChemMedChem

Country: Unknown

Publisher: Unknown

Language: N/A

Publication Details

Subject Category: Pharmacology

Available in Europe PMC: Yes

Available in PMC: Yes

PDF Available: No

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"crystallographic data centre via http://www ccdc cam ac uk/data_request/cif"

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"We thank A. C. Smith for technical assistance. This work was supported by Sterix Ltd., Wellcome Trust Programme Grant 082837 (to B.V.L.P.) and VIP funding."

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Last Updated: Aug 05, 2025