A monoclonal antibody raised against a thermo-stabilised β<sub>1</sub>-adrenoceptor interacts with extracellular loop 2 and acts as a negative allosteric modulator of a sub-set of β<sub>1</sub>-adrenoceptors expressed in stable cell lines.

Publication Year: 2017

DOI:
10.1016/j.bcp.2017.10.015

PMCID:
PMC5770334

PMID:
29102678

Journal Information

Full Title: Biochem Pharmacol

Abbreviation: Biochem Pharmacol

Country: Unknown

Publisher: Unknown

Language: N/A

Publication Details

Subject Category: Biochemistry

Available in Europe PMC: Yes

Available in PMC: Yes

PDF Available: No

Transparency Score
2/6
0.0% Transparent
Transparency Indicators
Click on green indicators to view evidence text
Core Indicators
Data Sharing
Code Sharing
Evidence found in paper:

"Conflict of interest AB, GC and CJH are shareholders in Heptares Therapeutics (part of the Sosei Group) and hold stock options in the Sosei Group. CJH is a consultant for Heptares Therapeutics. The remaining authors declare no conflict of interest."

Evidence found in paper:

"The work was supported by the Medical Research Council [grant numbers G0800006, MR/N020081/1], Heptares Therapeutics Ltd. and the University of Nottingham for financial support."

Protocol Registration
Open Access
Additional Indicators
Replication
Novelty Statement
Assessment Info

Tool: rtransparent

OST Version: N/A

Last Updated: Aug 05, 2025