From DC18 to MR07: A Metabolically Stable 4,4'-Oxybisbenzoyl Amide as a Low-Nanomolar Growth Inhibitor of P. falciparum.

Authors:
Bassanini I; Parapini S; Basilico N; Taramelli D; Romeo S.

Journal:
ChemMedChem

Publication Year: 2022

DOI:
10.1002/cmdc.202200355

PMCID:
PMC9827966

PMID:
36089546

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Journal Information

Full Title: ChemMedChem

Abbreviation: ChemMedChem

Country: Unknown

Publisher: Unknown

Language: N/A

Publication Details

Subject Category: Pharmacology

Available in Europe PMC: Yes

Available in PMC: Yes

PDF Available: No

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"Conflict of interest The authors declare no conflict of interest."

Evidence found in paper:

"This work was supported by Ministero dell'Istruzione, dell'Università e della Ricerca [PRIN 2015.4JRJPP_004] and University of Milan “Piano sostegno alla Ricerca, Linea 2 2018” ”to SR, Piano sostegno alla Ricerca, Linea 2 2020–2021 to NB and SP . We also thank the Immunohaematology and Transfusion Medicine Service, Department of Laboratory Medicine, ASST Grande Ospedale Metropolitano Niguarda (Milano) for providing erythrocytes for parasite cultures. We also thank Dr. Ugo Zanelli for pharmacokinetic studies. Open Access funding provided by Consiglio Nazionale delle Ricerche within the CRUI‐CARE Agreement."

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Last Updated: Aug 05, 2025