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High Target Homology Does Not Guarantee Inhibition: Aminothiazoles Emerge as Inhibitors of <i>Plasmodium falciparum</i>.
Johannsen S; Gierse RM; Krüger A; Edwards RL; Nanna V; Fontana A; Zhu D; Masini T; de Carvalho LP; Poizat M; Kieftenbelt B; Hodge DM; Alvarez S; Bunt D; Lacour A; Shams A; Meissner KA; de Souza EE; Dröge M; van Vliet B; den Hartog J; Hutter MC; Held J; Odom John AR; Wrenger C; Hirsch AKH.
ACS Infect Dis
(Unknown)
Published: 2024
Extracellular Vesicles in Malaria: Shedding Light on Pathogenic Depths.
ACS Infect Dis
(Unknown)
Published: 2024
Chelation of Mitochondrial Iron as an Antiparasitic Strategy.
Arbon D; Mach J; Čadková A; Sipkova A; Stursa J; Klanicová K; Machado M; Ganter M; Levytska V; Sojka D; Truksa J; Werner L; Sutak R.
ACS Infect Dis
(Unknown)
Published: 2024
Heterologous Sarbecovirus Receptor Binding Domains as Scaffolds for SARS-CoV-2 Receptor Binding Motif Presentation.
Hauser BM; Sangesland M; Lam EC; St Denis KJ; Sheehan ML; Vu ML; Cheng AH; Sordilla S; Lamson DT; Almawi AW; Balazs AB; Lingwood D; Schmidt AG.
ACS Infect Dis
(Unknown)
Published: 2024
Loratadine Combats Methicillin-Resistant <i>Staphylococcus aureus</i> by Modulating Virulence, Antibiotic Resistance, a…
Viering BL; Balogh H; Cox CF; Kirpekar OK; Akers AL; Federico VA; Valenzano GZ; Stempel R; Pickett HL; Lundin PM; Blackledge MS; Miller HB.
ACS Infect Dis
(Unknown)
Published: 2023
Quinoline Compounds Targeting the <i>c</i>-Ring of ATP Synthase Inhibit Drug-Resistant <i>Pseudomonas aeruginosa</i>.
Fraunfelter VM; Pugh BA; Williams APL; Ward KT; Jackson DO; Austin M; Ciprich JF; Dippy L; Dunford J; Edwards GN; Glass E; Handy KM; Kellogg CN; Llewellyn K; Nyberg KQ; Shepard SJ; Thomas C; Wolfe AL; Steed PR.
ACS Infect Dis
(Unknown)
Published: 2023
Shotgun Kinetic Target-Guided Synthesis Approach Enables the Discovery of Small-Molecule Inhibitors against Pathogenic …
Kassu M; Parvatkar PT; Milanes J; Monaghan NP; Kim C; Dowgiallo M; Zhao Y; Asakawa AH; Huang L; Wagner A; Miller B; Carter K; Barrett KF; Tillery LM; Barrett LK; Phan IQ; Subramanian S; Myler PJ; Van Voorhis WC; Leahy JW; Rice CA; Kyle DE; Morris J; Manetsch R.
ACS Infect Dis
(Unknown)
Published: 2023
Small-Molecule Antibiotic Drug Development: Need and Challenges.
ACS Infect Dis
(Unknown)
Published: 2023